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PARP Inhibitors

Cat.No. Product Name Information Publication Customer Review
S1060 Olaparib (AZD2281) Olaparib (AZD2281, KU0059436) is a selective inhibitor of PARP1 and PARP2 with IC50 of 5 nM and 1 nM, respectively. (23)
S1004 ABT-888 (Veliparib) ABT-888 (Veliparib, NSC 737664) is a potent inhibitor of PARP1 and PARP2 with Ki of 5.2 nM and 2.9 nM, respectively. (9)
S1098 Rucaparib (AG-014699 , PF-01367338) Rucaparib (AG-014699, PF-01367338) is an inhibitor of PARP with Ki of 1.4 nM. (3)
S1087 Iniparib (BSI-201) BSI-201 (Iniparib, SAR240550) is a PARP1 inhibitor. (1)
S2197 A-966492 A-966492 is a novel and potent inhibitor of PARP1 and PARP2 with Ki of 1 nM and 1.5 nM, respectively.
S2178 AG14361 AG14361 is a potent inhibitor of PARP1 with Ki of < 5 nM.
S1132 INO-1001 INO-1001 is a potent inhibitor of PARP with IC50 of 50 nM and a mediator of oxidant-induced myocyte dysfunction during reperfusion.
S7048 BMN 673 BMN 673 is a novel PARP inhibitor with IC50 of 0.58 nM.
S8038 UPF 1069 UPF 1069 is a selective PARP2 inhibitor with IC50 of 0.3 μM.
S2886 PJ34 PJ-34 is a potent PARP inhibitor with EC50 of 20 nM.
S2741 MK-4827 MK-4827 is an selective inhibitor of PARP1 and PARP2 with IC50 of 3.8 nM and 2.1 nM, respectively.