| Cat.No. |
Product Name |
Information |
Publication |
Customer Review |
| S2187 |
Avasimibe(CI-1011) |
Avasimibe inhibits ACAT and CYP2C9 with IC50 of 3.3 μM and 2.9 μM, respectively. |
|
|
| S2042 |
Cyproterone acetate |
Cyproterone acetate is an androgen receptor (AR) antagonist with IC50 of 7.1 nM. |
|
|
| S2757 |
TH-302 |
TH-302 is selective hypoxia-activated prodrug targeting hypoxic regions of solid tumors with IC50 of 19 nM. |
|
|
| S2803 |
Galeterone (TOK-001) |
Galeterone (TOK-001, VN/124-1) is a selective CYP17 inhibitor and androgen receptor (AR) antagonist with IC50 of 300 nM and 384 nM, respectively. |
|
|
| S1195 |
TAK-700 (Orteronel) |
TAK-700 (Orteronel) is a potent and highly selective rat and human 17,20-lyase inhibitor with IC50 of 54 nM and 38 nM, respectively. |
|
|
| S2526 |
Alizarin |
Alizarin strongly inhibits P450 isoform CYP1A1, CYP1A2 and CYP1B1 with IC50 of 6.2 μM, 10.0 μM and 2.7 μM, respectively. |
|
|
| S2921 |
PF-4981517 |
PF-4981517 is a potent and selective inhibitor of CYP3A4 (P450) with IC50 of 0.03 μM. |
|
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