Opioid receptors, which belong to G-protein-coupled super family, include mu-opioid receptor, delta-opioid receptor, and kappa-opioid receptor. Opioid receptors are receptor for opiate drugs. Opioid receptors can be found in the mammalian central nervous system and some other tissues, including the immune system. After opiate drugs binding to the specific receptor sites of opioid receptors, opioid receptors can executive function such as analgesia, sedation and so on.
| Cat.No. | Product Name | Information | Publication | Customer Review |
|---|---|---|---|---|
| S2722 | JTC-801 | JTC-801 is a selective opioid receptor-like1 (ORL1) receptor antagonist with IC50 of 94 nM. |
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| S1139 | ADL5859 HCl | ADL5859 HCl is a δ-opioid receptor agonist with Ki of 0.8 nM. |
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