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IGF-1R Inhibitors

Cat.No. Product Name Information Publication Customer Review
S1091 Linsitinib (OSI-906) OSI-906 (Linsitinib) is a selective inhibitor of IGF-1R and IR with IC50 of 35 nM and 75 nM, respectively. (2)
S1093 GSK1904529A GSK1904529A is a selective inhibitor of IGF-1R and IR with IC50 of 27 nM and 25 nM, respectively. (1)
S1088 NVP-ADW742 NVP-ADW742 is an IGF-1R inhibitor with IC50 of 0.17 μM.
S1034 NVP-AEW541 NVP-AEW541 is a potent inhibitor of IGF-1R with IC50 of 86 nM. (5)
S2703 GSK1838705A GSK1838705A is a potent inhibitor of IGF-1R, IR and ALK with IC50 of 2.0 nM, 1.6 nM and 0.5 nM, respectively
S1012 BMS-536924 BMS-536924 is an ATP-competitive IGF-1R and IR inhibitor with IC50 of 100 nM and 73 nM, respectively. (6)
S1124 BMS-754807 BMS-754807 is a potent and reversible inhibitor of IGF-1R/IR family kinases, inhibits IGF-1R, IR, Met, TrkA and TrkB with IC50 of 1.8 nM, 1.7 nM, 5.6 nM, 7.4 nM and 4.1 nM, respectively.
S8003 PQ 401 PQ 401 is an IGF-1R inhibitor with IC50 of <1 μM.
S1234 AG-1024 AG-1024 (Tyrphostin) is a specific IGF-1R and IR inhibitor with IC50 of 0.4 μM and 0.1 μM, respectively.