| Cat.No. |
Product Name |
Information |
Publication |
Customer Review |
| S2638 |
NU7441 (KU-57788) |
NU7441 is a highly potent and selective DNA-PK inhibitor with IC50 of 14 nM and also inhibits PI3K with IC50 of 5 μM.
|
 (1)
|
 (1)
|
| S1038 |
PI-103 |
PI-103 is a potent, ATP-competitive PI3K inhibitor of DNA-PK, p110α, mTORC1, PI3KC2β, p110δ, mTORC2, p110β, and p110γ with IC50 of 2 nM, 8 nM, 20 nM, 26 nM, 48 nM, 83 nM, 88 nM and 150 nM, respectively.
|
(5)
|
(4)
|
| S1205 |
PIK-75 |
PIK-75 is a selective and competitive inhibitor of p110α with IC50 of 5.8 nM and also potently inhibits DNA-PK with IC50 of 2 nM.
|
(1)
|
(2)
|
| S2893 |
NU7026 |
NU7026 is a DNA-PK inhibitor with IC50 of 0.23 μM.
|
|
|
| S2622 |
PP-121 |
PP-121 is a multi-target inhibitor of PDGFR, Hck, mTOR, VEGFR2, Src and Abl with IC50 of 2 nM, 8 nM, 10 nM, 12 nM, 14 nM and 18 nM, respectively, and also inhibits DNA-PK with IC50 of 60 nM.
|
|
(1)
|
